Bpsbioscience/Entacapone/27621-2/100 mg
商品编号:
27621-2
品牌:
bpsbioscience
市场价:
¥4800.00
美元价:
2880.00
联系Q Q:
3392242852
电话号码:
4000-520-616
电子邮箱:
info@ebiomall.com
商品介绍
MW: 305.3 Da
CAS Registry #: 130929-57-6
Formula: C14H15N3O5
Target: COMT
Description:
Entacapone is a second-generation catechol-O-methyltransferase (COMT) inhibitor
Synonym(s):
(E)-2-cyano-3-(3,4-dihydroxy-5-nitrophenyl)-N,N-diethylprop-2-enamide
Purity:
≥98% by HPLC
Biological Activity:
Entacapone potently inhibits rat liver total COMT with IC50 and Ki values of 20.1 nM and 10.7 nM respectively. The IC50 values of entacapone against rat liver soluble COMT (S-COMT) and rat liver membrane-bound COMT (MB-COMT) are 14.3 nM and 73.3 nM respectively.
Solubility:
Soluble in DMSO 61 mg/ml, water <1 mg/ml, ethanol 2 mg/ml
Storage / Stability:
Store at or below –20°C. Solid form is stable at least 12 months from date of receipt, when stored as directed. Do not store aqueous solutions for more than one day.
Reference(s):
Forsberg M, et al. J Pharmacol Exp Ther. 2003 Feb;304(2):498-506.
Scientific Category:
Methyltransferase Inhibitor
Product Type:
Inhibitor
Data shown is lot-specific. Contact us for specific information on other lots.
品牌介绍
bpsbioscience简介:为生命科学研究提供ELISA试剂盒(仅供科研)、抗体和抗原(仅供科研)、流式抗体,使您的检测结果更稳定可靠,用心服务科研。我公司国内总代理,华东地区代理bpsbioscience 专业经营进口胎牛血清、细胞因子、ELISA试剂盒、细胞、抗体、生物试剂、耗材、培养基、一抗、二抗、其产品吸附均匀,吸附性好,空白值低,孔底透明度高,代做ELISA实验等。