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3. Discoveryoffirst-in-classreversIBLedualsmallmoleculeinhibitorsagainstG9aandDNMTsinhematologicalmalignancies(2017)
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5.MolecularSimulationandActivityStudiesofOxametacinasanHDACInhibitor(2017)
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8. Design,synthesisandbiologicalevaluationofnovelhydroxamicacidbasedhistonedeacetylase6selectiveinhibitorsbearingphenylpyrazolscaffoldassurfacerecognitionmotif(2017)
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11. HDAC1-3inhibitorMS-275enhancesIL10expressioninRAW264.7macrophagesandreducescigarettesmoke-inducedairwayinflammationinmice (2017)
12. Novelanalogstargetinghistonedeacetylasesuppressaggressivethyroidcancercellgrowthandinducere-differentiation(2015)
13.Design,synthesis,3Dpharmacophore,QSAR,anddockingstudiesofcarboxylicacidderivativesasHistoneDeacetylaseinhibitorsandcytotoxicagents(2014)
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15.Kineticmethodforthelarge-scaleanalysisofthebindingmechanismofhistonedeacetylaseinhibitors(2014)
16.ThermodynamicsofligandbindingtohistonedeacetylaselikeamidohydrolasefromBordetella/Alcaligenes(2014)
17.AselectiveHDAC1/2inhibitormodulateschromatinandgeneexpressioninbrainandaltersmousebehaviorintwomood-relatedtests(2013)
18.Crebinostat:anovelcognitiveenhancerthatinhibitshistonedeacetylaseactivityandmodulateschromatin-mediatedneuroplasticity(2013)
19.HighlyligandefficientandselectiveN-2-(Thioethyl)picolinamidehistonedeacetylaseinhibitorsinspiredbythenaturalproductpsammaplinA(2013)
20.Potenthistonedeacetylaseinhibitorsderivedfrom4-(aminomethyl)-N-hydroxybenzamidewithhighselectivityfortheHDAC6isoform(2013)
21.SantacruzamateA,apotentandselectivehistonedeacetylaseinhibitorfromthePanamanianmarinecyanobacteriumcf.Symplocasp(2013)
22.ThioesterderivativesofthenaturalproductpsammaplinAaspotenthistonedeacetylaseinhibitors(2013)
