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ApplicationReference(s):
1. SelectivityandKineticRequirementsofHDACInhibitorsasProgranulinEnhancersforTreatingFrontotemporalDementia(2017)
2. AnazumamideCanaloguewithoutthezinc-bindingfunctionality(2017)
3. MolecularSimulationandActivityStudiesofOxametacinasanHDACInhibitor(2017)
4. Impactofbindingmechanismonselectiveinhibitionofhistonedeacetylaseisoforms(2017)
5. Design,synthesisandBIOLOGicalevaluationofnovelhydroxamicacidbasedhistonedeacetylase6selectiveinhibitorsbearingphenylpyrazolscaffoldassurfacerecognitionmotif(2017)
6.IdentificationofhistonedeacetylaseinhibitorswithbenzoylhydrazidescaffoldthatselectivelyinhibitclassIhistonedeacetylases(2015)
7.MechanismofActionof2-AminobenzamideHDACInhibitorsinReversingGeneSilencinginFriedreich"sAtaxia(2015)
8.Design,synthesis,3Dpharmacophore,QSAR,anddockingstudiesofcarboxylicacidderivativesasHistoneDeacetylaseinhibitorsandcytotoxicagents(2014)
9.DiscoveryofasmallmoleculeagoNISTofphosphatidylinositol3-kinasep110αthatreactivateslatentHIV-1(2014)
10.AchimericSERM-histonedeacetylaseinhibitorapproachtobreastcancertherapy(2014)
11.InVivoImagingofHistoneDeacetylases(HDACs)intheCentralNervousSystemandMajorPeripheralOrgans(2014)
12.SelectiveHDACInhibitionfortheDisruptionofLatentHIV-1Infection(2014)
13.ClassIHDACimagingusing[(3)H]CI-994autorADIography(2013)
14.Crebinostat:anovelcognitiveenhancerthatinhibitshistonedeacetylaseactivityandmodulateschromatin-mediatedneuroplasticity(2013)
15.FDG-PETimagingrevealslocalbrainglucoseutilizationisalteredbyclassIhistonedeacetylaseinhibitors(2013)
16.HighlyligandefficientandselectiveN-2-(Thioethyl)picolinamidehistonedeacetylaseinhibitorsinspiredbythenaturalproductpsammaplinA(2013)
17.ImagingepigeneticregulationbyhistonedeacetylasesinthebrainusingPET/MRIwith¹⁸F-FAHA(2013)
18.Structuralbasisfortheinhibitionofhistonedeacetylase8(HDAC8),akeyepigeneticplayerinthebloodflukeSchistosomamansoni(2013)